De novo design of α-helical lipopeptides targeting viral fusion proteins: a promising strategy for relatively broad-spectrum antiviral drug discovery

C Wang, L Zhao, S Xia, T Zhang, R Cao… - Journal of medicinal …, 2018 - ACS Publications
C Wang, L Zhao, S Xia, T Zhang, R Cao, G Liang, Y Li, G Meng, W Wang, W Shi, W Zhong…
Journal of medicinal chemistry, 2018ACS Publications
Class I enveloped viruses share similarities in their apparent use of a hexameric coiled-coil
assembly to drive the merging of virus and host cell membranes. Inhibition of coiled coil-
mediated interactions using bioactive peptides that replicate an α-helical chain from the viral
fusion machinery has significant antiviral potential. Here, we present the construction of a
series of lipopeptides composed of a de novo heptad repeat sequence-based α-helical
peptide plus a hydrocarbon tail. Promisingly, the constructs adopted stable α-helical …
Class I enveloped viruses share similarities in their apparent use of a hexameric coiled-coil assembly to drive the merging of virus and host cell membranes. Inhibition of coiled coil-mediated interactions using bioactive peptides that replicate an α-helical chain from the viral fusion machinery has significant antiviral potential. Here, we present the construction of a series of lipopeptides composed of a de novo heptad repeat sequence-based α-helical peptide plus a hydrocarbon tail. Promisingly, the constructs adopted stable α-helical conformations and exhibited relatively broad-spectrum antiviral activities against Middle East respiratory syndrome coronavirus (MERS-CoV) and influenza A viruses (IAVs). Together, these findings reveal a new strategy for relatively broad-spectrum antiviral drug discovery by relying on the tunability of the α-helical coiled-coil domains present in all class I fusion proteins and the amphiphilic nature of the individual helices from this multihelix motif.
ACS Publications